Dacheux Mélanie, Sinou Véronique, Payré Christine, Jeammet Louise, Parzy Daniel, Grellier Philippe, Deregnaucourt Christiane & Lambeau Gérard, août 2019 — Antimalarial Activity of Human Group IIA Secreted Phospholipase A _{\textrm{2}} in Relation to Enzymatic Hydrolysis of Oxidized Lipoproteins. Infection and Immunity vol. 87, n° 11,
ISSN
0019-9567, 1098-5522
https://dx.doi.org/10.1128/IAI.00556-19
Holota Serhii, Kryshchyshyn Anna, Derkach Halyna, Trufin Yaroslava, Demchuk Inna, Gzella Andrzej, Grellier Philippe & Lesyk Roman, mai 2019 — Synthesis of 5-enamine-4-thiazolidinone derivatives with trypanocidal and anticancer activity. Bioorganic Chemistry vol. 86, , p. 126-136
ISSN
00452068
https://dx.doi.org/10.1016/j.bioorg.2019.01.045
Marozienė Audronė, Lesanavičius Mindaugas, Davioud-Charvet Elisabeth, Aliverti Alessandro, Grellier Philippe, Šarlauskas Jonas & Čėnas Narimantas, décembre 2019 — Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase. Molecules vol. 24, n° 24, p. 4509
ISSN
1420-3049
https://dx.doi.org/10.3390/molecules24244509
Kryshchyshyn Anna, Kaminskyy Danylo, Karpenko Oleksandr, Gzella Andrzej, Grellier Philippe & Lesyk Roman, juillet 2019 — Thiazolidinone/thiazole based hybrids – New class of antitrypanosomal agents. European Journal of Medicinal Chemistry vol. 174, , p. 292-308
ISSN
02235234
https://dx.doi.org/10.1016/j.ejmech.2019.04.052
Motta Flávia Nader, Azevedo Clênia dos Santos, Neves BeatrizPereira, Araújo Carla Nunes de, Grellier Philippe, Santana Jaime Martins de & Bastos Izabela Marques Dourado, décembre 2019 — Oligopeptidase B, a missing enzyme in mammals and a potential drug target for trypanosomatid diseases. Biochimie vol. 167, , p. 207-216
ISSN
03009084
https://dx.doi.org/10.1016/j.biochi.2019.10.006
Terzic Vida, Pousse Guillaume, Méallet-Renault Rachel, Grellier Philippe & Dubois Joëlle, juillet 2019 — Dibenzocyclooctynes: Effect of Aryl Substitution on Their Reactivity toward Strain-Promoted Alkyne–Azide Cycloaddition. The Journal of Organic Chemistry vol. 84, n° 13, p. 8542-8551
ISSN
0022-3263, 1520-6904
https://dx.doi.org/10.1021/acs.joc.9b00895