Bounaadja Lotfi, Schmitt Marjorie, Albrecht Sébastien, Mouray Elisabeth, Tarnus Céline & Florent Isabelle, December 2017 — Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo. Malaria Journal vol. 16, n° 1,
ISSN
1475-2875
https://dx.doi.org/10.1186/s12936-017-2032-4
Pascual Isel, Valiente Pedro A., García Gabriela, Valdés-Tresanco Mario E., Arrebola Yarini, Díaz Lisset, Bounaadja Lotfi, Uribe Rosa María, Pacheco Mae Chappé, Florent Isabelle & Charli Jean-Louis, November 2017 — Discovery of novel non-competitive inhibitors of mammalian neutral M1 aminopeptidase (APN). Biochimie vol. 142, , p. 216-225
ISSN
03009084
https://dx.doi.org/10.1016/j.biochi.2017.09.015
González-Bacerio Jorge, Maluf Sarah El Chamy, Méndez Yanira, Pascual Isel, Florent Isabelle, Melo Pollyana M.S., Budu Alexandre, Ferreira Juliana C., Moreno Ernesto, Carmona Adriana K., Rivera Daniel G., Alonso del Rivero Maday & Gazarini Marcos L., September 2017 — KBE 009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library. Bioorganic \& Medicinal Chemistry vol. 25, n° 17, p. 4628-4636
ISSN
09680896
https://dx.doi.org/10.1016/j.bmc.2017.06.047